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Michael W. Crowder

University System of Ohio

42H指数
179论文数
5.6K被引数
收录论文 63
发表时间
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Inhibitor Affinity Differs among Clinical Variants of IMP Metallo-β-Lactamases: Analysis and Implications for Inhibitor Design抑制剂亲和力在不同临床类型的IMP金属-β-内酰胺酶之间存在差异:分析与抑制剂设计的意义
err2025-07-24
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PREAI
errCaitlyn A. Thomas; John Paul Alao; Thomas Smisek; Zishuo Cheng; Christopher R. Bethel; Kundi Yang; Ikponwmosa Obaseki; Richard C. Page; Robert A. Bonomo; Peter Oelschlaeger; Walter Fast; Andrea N. Kravats; Michael W. Crowder
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Machine Learning Models Identify Inhibitors of New Delhi Metallo-β-lactamase
err2024-05-10
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errCheng, Zishuo; Aitha, Mahesh; Thomas, Caitlyn A.; Sturgill, Aidan; Fairweather, Mitch; Hu, Amy; Bethel, Christopher R.; Rivera, Dann D.; Dranchak, Patricia; Thomas, Pei W.; Li, Han; Feng, Qi; Tao, Kaicheng; Song, Minshuai; Sun, Na; Wang, Shuo; Silwal, Surendra Bikram; Page, Richard C.; Fast, Walt; Bonomo, Robert A.; Weese, Maria; Martinez, Waldyn; Inglese, James; Crowder, Michael W.
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The directed evolution of NDM-1NDM-1的定向进化
err2023-11-15
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errThomas, Caitlyn A.; Cheng, Zishuo; Bethel, Christopher R.; Hujer, Andrea M.; Sturgill, Aidan M.; Onuoha, Kelechi; Page, Richard C.; Bonomo, Robert A.; Crowder, Michael W.; Tamma, Pranita D.
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Taxifolin as a Metallo-β-Lactamase Inhibitor in Combination with Augmentin against Verona Imipenemase 2 Expressing Pseudomonas aeruginosa
err2023-10-28
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errBenin, Bogdan M.; Hillyer, Trae; Crugnale, Aylin S.; Fulk, Andrew; Thomas, Caitlyn A.; Crowder, Michael W.; Smith, Matthew A.; Shin, Woo Shik
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Characterizing bourbon whiskey via the combination of LC-MS and GC-MS based molecular fingerprinting
err2023-10-01
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PREAI
errXu, Rui; Chen, Li; Zhang, Huan; Crowder, Michael W.; Zhu, Jiangjiang
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Profiling bourbons based on congener concentrations
err2023-01-01
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PREAI
errZhang, Huan; Johnson, Eric C.; Carroll, Anne; Pryor, Cecily; Howe, Kenneth; Kramer, Ryan; Rajesh, Naik; Meyer, Emily; Shurina, Ben; Kumarage, Nuwanthika; Yang, Kundi; Kennedy, Michael A.; Crowder, Michael W.
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Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates
err2022-11-30
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errLegru, Alice; Verdirosa, Federica; Vo-Hoang, Yen; Tassone, Giusy; Vascon, Filippo; Thomas, Caitlyn A.; Sannio, Filomena; Corsica, Giuseppina; Benvenuti, Manuela; Feller, Georges; Coulon, Remi; Marcoccia, Francesca; Devente, Savannah Rowane; Bouajila, Ezeddine; Piveteau, Catherine; Leroux, Florence; Deprez-Poulain, Rebecca; Deprez, Benoit; Licznar-Fajardo, Patricia; Crowder, Michael W.; Cendron, Laura; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-Francois; Gavara, Laurent
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Discovery of an Effective Small-Molecule Allosteric Inhibitor of New Delhi Metallo-β-lactamase (NDM)
err2022-03-30
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PREAI
errThomas, Pei W.; Cho, Eun Jeong; Bethel, Christopher R.; Smisek, Thomas; Ahn, Yeong-Chan; Schroeder, John M.; Thomas, Caitlyn A.; Dalby, Kevin N.; Beckham, Josh T.; Crowder, Michael W.; Bonomo, Robert A.; Fast, Walter
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1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity
err2021-12-01
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errLegru, Alice; Verdirosa, Federica; Hernandez, Jean-Francois; Tassone, Giusy; Sannio, Filomena; Benvenuti, Manuela; Conde, Pierre-Alexis; Bossis, Guillaume; Thomas, Caitlyn A.; Crowder, Michael W.; Dillenberger, Melissa; Becker, Katja; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Gavara, Laurent
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Fragment-based screening and hit-based substructure search: Rapid discovery of 8-hydroxyquinoline-7-carboxylic acid as a low-cytotoxic, nanomolar metallo β-lactamase inhibitor
err2021-07-23
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PREAI
errShin, Woo Shik; Nguyen, Megin E.; Bergstrom, Alexander; Jennings, Isabella R.; Crowder, Michael W.; Muthyala, Ramaiah; Sham, Yuk Yin
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Spectroscopic and biochemical characterization of metallo-8-lactamase IMP-1 with dicarboxylic, sulfonyl, and thiol inhibitors
err2021-06-01
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errZhang, Huan; Yang, Kundi; Cheng, Zishuo; Thomas, Caitlyn; Steinbrunner, Abbie; Pryor, Cecily; Vulcan, Maya; Kemp, Claire; Orea, Diego; Paththamperuma, Chathura; Chen, Allie Y.; Cohen, Seth M.; Page, Richard C.; Tierney, David L.; Crowder, Michael W.
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Visualizing the Dynamic Metalation State of New Delhi Metallo-β-actamase-1 in Bacteria Using a Reversible Fluorescent Probe
err2021-05-26
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errMehta, Radhika; Rivera, Dann D.; Reilley, David J.; Tan, Dominique; Thomas, Pei W.; Hinojosa, Abigail; Stewart, Alesha C.; Cheng, Zishuo; Thomas, Caitlyn A.; Crowder, Michael W.; Alexandrova, Anastassia N.; Fast, Walter; Que, Emily L.
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Carbapenem Use Is Driving the Evolution of Imipenemase 1 Variants
err2021-03-18
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errCheng, Zishuo; Bethel, Christopher R.; Thomas, Pei W.; Shurina, Ben A.; Alao, John-Paul; Thomas, Caitlyn A.; Yang, Kundi; Marshall, Steven H.; Zhang, Huan; Sturgill, Aidan M.; Kravats, Andrea N.; Page, Richard C.; Fast, Walter; Bonomo, Robert A.; Crowder, Michael W.
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Probing the mechanisms of inhibition for various inhibitors of metallo-β-lactamases VIM-2 and NDM-1
err2020-09-01
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PREAI
errThomas, Caitlyn A.; Cheng, Zishuo; Yang, Kundi; Hellwarth, Elle; Yurkiewicz, Cole J.; Baxter, Faith M.; Fullington, Sarah A.; Klinsky, Spencer A.; Otto, Jen L.; Chen, Allie Y.; Cohen, Seth M.; Crowder, Michael W.
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Iminodiacetic Acid as a Novel Metal-Binding Pharmacophore for New Delhi Metallo-β-lactamase Inhibitor Development
err2020-05-07
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errChen, Allie Y.; Thomas, Caitlyn A.; Thomas, Pei W.; Yang Kundi; Cheng Zishuo; Fast, Walter; Crowder, Michael W.; Cohen, Seth M.
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Elusive structural changes of New Delhi metallo-β-lactamase revealed by ultraviolet photodissociation mass spectrometry
err2020-01-01
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errMehaffey, M. Rachel; Ahn, Yeong-Chan; Rivera, Dann D.; Thomas, Pei W.; Cheng, Zishuo; Crowder, Michael W.; Pratt, R. F.; Fast, Walter; Brodbelt, Jennifer S.
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A Single Salt Bridge in VIM-20 Increases Protein Stability and Antibiotic Resistance under Low-Zinc Conditions
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IF4.7
err2019-12-24
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errCheng, Zishuo; Shurina, Ben A.; Bethel, Christopher R.; Thomas, Pei W.; Marshall, Steven H.; Thomas, Caitlyn A.; Yang, Kundi; Kimble, Robert L.; Montgomery, Jonathan S.; Orischak, Matthew G.; Miller, Callie M.; Tennenbaum, Jordan L.; Nix, Jay C.; Tierney, David L.; Fast, Walter; Bonomo, Robert A.; Page, Richard C.; Crowder, Michael W.
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Investigation of Dipicolinic Acid Isosteres for the Inhibition of Metallo-β-Lactamases
err2019-05-24
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errChen, Allie Y.; Thomas, Pei W.; Cheng, Zishuo; Xu, Nasa Y.; Tierney, David L.; Crowder, Michael W.; Fast, Walter; Cohen, Seth M.
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