Prem N. Yadav - Publications, H-index & Citations

Prem N. Yadav

csir - central drug research institute (cdri)

33H指数

112论文数

3.4K被引数

收录论文 44

发表时间

Modular synthesis and bioevaluation of novel fused-β-carbolines as kappa opioid receptor modulators 新型杂环β-咔啉的模块化合成与生物活性评价及其作为κ阿片受体调节剂的应用

European Journal of Medicinal Chemistry

IF5.9

2026-07-01

PREAI

Ghosh, Aritra; Dash, Manish K.; Shukla, Nupoor; Pandey, Ghanshyam; Siddiqi, Mohammad I.; Chakradhar, J. V. U. S.; Singh, Yuvraj; Kant, Ruchir; Yadav, Prem N.; Batra, Sanjay

Towards next-generation 5-hydroxytryptamine 2C receptor modulators: Greener synthesis and evaluation of novel isocoumarin derivatives as PAAMs of 5-HT2CR 面向下一代5-羟色胺2C受体调节剂：绿色合成与新型异香豆素衍生物作为5-HT2CR PAAMs的评估

Bioorganic Chemistry

IF4.7

2025-11-24

PREAI

Kaushik Sarkar; Deepesh Biswas; B. Yogi Sreenivas; Rapaka Naimisha; Navneet Bung; Sedam Sai Madhuri; Raghavender Medishetti; Arijit Roy; Varadaraj Bhat Giliyaru; Prem N. Yadav; Kiranam Chatti; Srinivas Oruganti; Parimal Misra; Manojit Pal

Novel bis(triazole) analogues as selective TGR5 agonists with anti-diabesity effects 新型双三氮唑类似物作为选择性TGR5激动剂，具有抗糖尿病和肥胖的双重效果

Bioorganic Chemistry

IF4.7

2025-11-22

PREAI

Anchal Saxena; Devanshu Kaushik; Boda Arun Kumar; Shivam Rathaur; Diwan Chand; Kinshuk R. Srivastava; Jiaur R. Gayen; Prem N. Yadav; Nayan Ghosh

Synthesis and Evaluation of Novel Aza-Aromatics as Dual 5-HT2A and 5-HT2C Receptor Agonists 新型氮杂芳香族化合物的合成与评价：作为5-HT2A和5-HT2C受体双重激动剂

ACS MEDICINAL CHEMISTRY LETTERS

IF4

2025-11-01

PREAI

Adhikari, Amit Singh; Yadav, Annu; Pandit, Soumen; Kumar, Suresh; Pandey, Vinay Kumar; Maurya, Arvind Kumar; Umrao, Deepmala; Chand, Diwan; Maity, Debalina; Gayen, Jiaur R.; Srivastava, Kinshuk Raj; Yadav, Prem N.; Majumdar, Nilanjana

Editorial Expression of Concern: Atrial natriuretic factor receptor guanylate cyclase signaling: new ATP-regulated transduction motif 编者按：关注心房利钠因子受体鸟苷酸环化酶信号传导：新的ATP调控转导模式

Molecular and Cellular Biochemistry

IF3.7

2025-08-30

PREAI

Teresa Duda; Shashank Bharill; Ireneusz Wojtas; Prem Yadav; Ignacy Gryczynski; Zygmunt Gryczynski; Rameshwar K. Sharma

Neuronal Membrane-Coated Mesoporous Ceria Nanoparticles for Blood-Brain Barrier Crossing and Mitigation of Neurodegeneration 神经元膜包覆的介孔二氧化铈纳米颗粒用于血脑屏障穿越和神经退行性病变的缓解

ACS APPLIED NANO MATERIALS

IF5.5

2025-05-02

PREAI

Rana, R; Tripathi, S; Mishra, K; Yadav, PK; Yadav, PN; Chourasia, MK

Kappa Opioid Receptor Activation Induces Epigenetic Silencing of Brain-Derived Neurotropic Factor via HDAC5 in Depression

ACS CHEMICAL NEUROSCIENCE

IF3.9

2024-08-27

PREAI

Yadav, Anubhav; Dogra, Shalini; Boda, Arun Kumar; Kumari, Poonam; Kumar, Ajeet; Dash, Manish K.; Yadav, Prem N.

An amide to thioamide substitution improves the permeability and bioavailability of macrocyclic peptides

NATURE COMMUNICATIONS

IF15.7

2023-09-28

OAAI

Ghosh, Pritha; Raj, Nishant; Verma, Hitesh; Patel, Monika; Chakraborti, Sohini; Khatri, Bhavesh; Doreswamy, Chandrashekar M.; Anandakumar, S. R.; Seekallu, Srinivas; Dinesh, M. B.; Jadhav, Gajanan; Yadav, Prem Narayan; Chatterjee, Jayanta

Molecular insights into intrinsic transducer-coupling bias in the CXCR4-CXCR7 system

NATURE COMMUNICATIONS

IF15.7

2023-08-09

OAAI

Sarma, Parishmita; Carino, Carlo Marion C.; Seetharama, Deeksha; Pandey, Shubhi; Dwivedi-Agnihotri, Hemlata; Rui, Xue; Cao, Yubo; Kawakami, Kouki; Kumari, Poonam; Chen, Yu-Chih; Luker, Kathryn E.; Yadav, Prem N.; Luker, Gary D.; Laporte, Stephane A.; Chen, Xin; Inoue, Asuka; Shukla, Arun K.

Recent Advancements in Nanocarrier-assisted Brain Delivery of Phytochemicals Against Neurological Diseases

NEUROCHEMICAL RESEARCH

IF3.8

2023-06-06

PREAI

Mishra, Keerti; Rana, Rafquat; Tripathi, Shourya; Siddiqui, Shumaila; Yadav, Pavan K.; Yadav, Prem N.; Chourasia, Manish K.

Molecular determinants associated with temporal succession of SARS-CoV-2 variants in Uttar Pradesh, India

FRONTIERS IN MICROBIOLOGY

IF4.5

2023-02-01

OAAI

Pal, Smita; Mehta, Poonam; Pandey, Ankita; Ara, Anam; Ghoshal, Ujjala; Ghoshal, Uday C. C.; Pandey, Rajesh; Tripathi, Raj Kamal; Yadav, Prem N. N.; Ravishankar, Ramachandran; Kundu, Tapas K. K.; Rajender, Singh

Copper-Catalyzed Oxidative [3+2]-Annulation of Quinoxalin2(1H)-one with Oxime Esters toward Functionalized Pyrazolo[1,5-a]quinoxalin-4(5H)-ones as Opioid Receptor Modulators

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2022-05-19

PREAI

Yadav, Anamika; Yadav, Anubhav; Tripathi, Shashank; Dewaker, Varun; Kant, Ruchir; Yadav, Prem Narayan; Srivastava, Ajay Kumar

Synthesis and Assessment of Fused β-Carboline Derivatives as Kappa Opioid Receptor Agonists

CHEMMEDCHEM

IF3.4

2021-03-18

PREAI

Yadav, Veena D.; Kumar, Lalan; Kumari, Poonam; Kumar, Sakesh; Singh, Maninder; Siddiqi, Mohammad I.; Yadav, Prem N.; Batra, Sanjay

Novel Tetrahydroquinazolinamines as Selective Histamine 3 Receptor Antagonists for the Treatment of Obesity

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2019-04-18

PREAI

Kumar, Ajeet; Pasam, Venkata Reddy; Thakur, Ravi Kumar; Singh, Maninder; Singh, Kartikey; Shukla, Mahendra; Yadav, Anubhav; Dogra, Shalini; Sona, Chandan; Umrao, Deepmala; Jaiswal, Swati; Ahmad, Hafsa; Rashid, Mamunur; Singh, Sandeep K.; Wahajuddin, Muhammad; Dwivedi, Anil Kumar; Siddiq, Mohammad Imran; Lal, Jawahar; Tripathi, Rama Pati; Yadav, Prem N.

Chronic histamine 3 receptor antagonism alleviates depression like conditions in mice via modulation of brain-derived neurotrophic factor and hypothalamus-pituitary adrenal axis

PSYCHONEUROENDOCRINOLOGY

IF3.6

2019-03-01

PREAI

Kumar, Ajeet; Dogra, Shalini; Sona, Chandan; Umrao, Deepmala; Rashid, Mamunur; Singh, Sandeep K.; Wahajuddin, Muhammad; Yadav, Prem N.

Identification of dual role of piperazine-linked phenyl cyclopropyl methanone as positive allosteric modulator of 5-HT2C and negative allosteric modulator of 5-HT2B receptors

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2019-02-01

PREAI

Singh, Kartikey; Sona, Chandan; Ojha, Vikash; Singh, Maninder; Mishra, Ankita; Kumar, Ajeet; Siddiqi, Mohammad Imran; Tripathi, Rama P.; Yadav, Prem N.

Docosahexaenoic acid modulates brain-derived neurotrophic factor via GPR40 in the brain and alleviates diabesity-associated learning and memory deficits in mice

NEUROBIOLOGY OF DISEASE

IF5.6

2018-10-01

PREAI

Sona, Chandan; Kumar, Ajeet; Dogra, Shalini; Kumar, Boda Arun; Umrao, Deepmala; Yadav, Prem N.

Identification of novel β-lactams and pyrrolidinone derivatives as selective Histamine-3 receptor (H3R) modulators as possible anti-obesity agents (vol 152, pg 148, 2018)

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2018-08-01

PREAI

Ghoshal, Anirban; Kumar, Ajeet; Yugandhar, Doddapaneni; Sona, Chandan; Kuriakose, Sunu; Nagesh, Kommu; Rashid, Mamunur; Singh, Sandeep K.; Wahajuddin, Muhammad; Yadav, Prem N.; Srivastava, Ajay K.

Discovery of coumarin-dihydroquinazolinone analogs as niacin receptor 1 agonist with in-vivo anti-obesity efficacy

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2018-05-01

PREAI

Singh, L. Ravithej; Kumar, Ajeet; Upadhyay, Akanksha; Gupta, Sampa; Palanati, Gopala Reddy; Sikka, Kamakshi; Siddiqi, Mohammad Imran; Yadav, Prem N.; Sashidhara, Koneni V.

Identification of novel β-lactams and pyrrolidinone derivatives as selective Histamine-3 receptor (H3R) modulators as possible anti-obesity agents

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2018-05-01

PREAI

Ghoshal, Anirban; Kumar, Ajeet; Yugandhar, Doddapaneni; Sona, Chandan; Kuriakose, Sunu; Nagesh, Kommu; Rashid, Mamunur; Singh, Sandeep K.; Wahajuddin, Muhammad; Yadav, Prem N.; Srivastava, Ajay K.

研究方向