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张

张岩 (Yan Zhang)

Virginia Commonwealth University

35H指数
238论文数
4.8K被引数
收录论文 105
发表时间
Structural Determinants of μ-Opioid Receptor Antagonism and Respiratory Liability in Phenylfentanyl Analogues苯基哌替啶类似物中μ-阿片受体拮抗作用和呼吸副作用的结构决定因素
err2026-04-30
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errEnnian Li; Balaji S. Kale; Abeje A. Silte; Rui Lyu; Neha Upadhyay; Logan T. Neel; Ahmed Reda; Huiqun Wang; William L. Dewey; Piyusha P. Pagare; Yan Zhang
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Investigating the Landscape of C6-Azaindole Side Chain on the Epoxymorphinan Skeleton via the Nitrogen Walk Concept: A Strategy to Enhance Drug-Like Properties
err2026-01-22
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errLogan Neel; Hongguang Ma; Ahmed Reda; Mengchu Li; Rachael Flammia; Samuel Woodard; James C. Gillespie; Dana E. Selley; William L. Dewey; Piyusha P. Pagare; Yan Zhang
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Design, Syntheses, and Pharmacological Evaluations of Core Ring Expanded Fentanyl Analogues as Potential Counteracting Agents Against Fentanyl Induced Respiratory Depression
err2025-11-01
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PREAI
errSilte, Abeje A.; Li, Ennian; Kale, Balaji S.; Neel, Logan; Upadhyay, Neha; Flammia, Rachael; Lyu, Rui; St Onge, Celsey M.; Reda, Ahmed; Woodard, Samuel; Gillespie, James C.; Kim, Daniel; Selley, Dana E.; Dewey, William L.; Pagare, Piyusha P.; Zhang, Yan
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Systematic Structure-Activity Relationship Study of Nalfurafine Analogues toward Development of Potentially Nonaddictive Pain Management Treatments
err2024-05-30
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errSt. Onge, Celsey M.; Pagare, Piyusha P.; Zheng, Yi; Arriaga, Michelle; Stevens, David L.; Mendez, Rolando E.; Poklis, Justin L.; Halquist, Matthew S.; Selley, Dana E.; Dewey, William L.; Banks, Matthew L.; Zhang, Yan
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NCP, a Dual Kappa and Mu Opioid Receptor Agonist, Is a Potent Analgesic Against Inflammatory Pain without Reinforcing or Aversive Properties
err2024-04-01
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errHuang, Peng; Ho, Conrad K.; Cao, Danni; Inan, Saadet; Rawls, Scott M.; Li, Mengchu; Huang, Boshi; Pagare, Piyusha P.; Townsend, E. Andrew; Poklis, Justin L.; Halquist, Matthew S.; Banks, Matthew; Zhang, Yan; Liu-Chen, Lee-Yuan
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Novel PROTAC probes targeting KDM3 degradation to eliminate colorectal cancer stem cells through inhibition of Wnt/β-catenin signaling
err2024-01-01
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errZaman, Shadid U.; Pagare, Piyusha P.; Ma, Hongguang; Hoyle, Rosalie G.; Zhang, Yan; Li, Jiong
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METTL3-mediated m6A RNA methylation was involved in aluminum-induced neurotoxicityMETTL3-mediated m6A RNA甲基化参与铝诱导的神经毒性
err2024-01-01
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errYang, Lingling; Chen, Liping; Li, Wenxue; Zhang, Yan; Yang, Guangyu; Huang, Bing; Cen, Yufang; Wang, Huiqi; Yang, Xueqin; Lin, Fangqin; Pang, Yaqin; Qi, Guangzi
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Molecular Pharmacology Profiling of Phenylfentanil and Its Analogues to Understand the Putative Involvement of an Adrenergic Mechanism in Fentanyl-Induced Respiratory Depression
err2023-12-29
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PREAI
errLi, Mengchu; Pagare, Piyusha P.; Ma, Hongguang; St Onge, Celsey M.; Mendez, Rolando E.; Gillespie, James C.; Stevens, David L.; Dewey, William L.; Selley, Dana E.; Zhang, Yan
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A cutting-edge strategy for spinal cord injury treatment: resident cellular transdifferentiation
err2023-08-30
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errFang, Yu-Ming; Chen, Wei-Can; Zheng, Wan-Jing; Yang, Yu-Shen; Zhang, Yan; Chen, Xin-Li; Pei, Meng-Qin; Lin, Shu; He, He-Fan
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Quantitative assessment of the in-vitro binding kinetics of antisickling aromatic aldehydes with hemoglobin A: A universal HPLC-UV/Vis method to quantitate Schiff-base adduct formation
err2023-01-01
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errXu, Xiaomeng; Ghatge, Mohini S.; Huang, Boshi; Alghamdi, Ahmed; Wang, Huiqun; Pierce, Daniel; Abdulmalik, Osheiza; Zhang, Yan; Safo, Martin K.; Venitz, Juergen
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Structural Alterations of the Address Moiety of NAN Leading to the Discovery of a Novel Opioid Receptor Modulator with Reduced hERG Toxicity
err2022-12-20
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errMa, Hongguang; Pagare, Piyusha P.; Li, Mengchu; Neel, Logan T.; Mendez, Rolando E.; Gillespie, James C.; Stevens, David L.; Dewey, William L.; Selley, Dana E.; Zhang, Yan
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研究方向

G蛋白偶联受体和信号转导研究基于受体和信号转导的天然产物药物筛选免疫抗炎活性天然产物的发现及机制研究