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Angelo Carotti

universita degli studi di bari aldo moro

50H-index
365Paper Count
8.4KCitation Count
Published Papers 103
Publication Date
Thioxanthenone-based derivatives as multitarget therapeutic leads for Alzheimer's disease
err2023-03-01
err14
errOAAI
errTonelli, Michele; Catto, Marco; Sabate, Raimon; Francesconi, Valeria; Laurini, Erik; Pricl, Sabrina; Pisani, Leonardo; Miniero, Daniela Valeria; Liuzzi, Grazia Maria; Gatta, Elena; Relini, Annalisa; Gavin, Rosalina; Rio, Jose Antonio Del; Sparatore, Fabio; Carotti, Angelo
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17β-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer
err2021-11-18
err5
errOAAI
errGargano, Emanuele M.; Mohamed, Abdelrahman; Abdelsamie, Ahmed S.; Mangiatordi, Giuseppe F.; Drzewiecka, Hanna; Jagodzinski, Pawel P.; Mazzini, Arcangela; van Koppen, Chris J.; Laschke, Matthias W.; Nicolotti, Orazio; Carotti, Angelo; Marchais-Oberwinkler, Sandrine; Hartmann, Rolf W.; Frotscher, Martin
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Coumarin: A Natural, Privileged and Versatile Scaffold for Bioactive Compounds
err2018-01-27
err484
errOAAI
errStefanachi, Angela; Leonetti, Francesco; Pisani, Leonardo; Catto, Marco; Carotti, Angelo
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Potent inhibitors of human LAT1 (SLC7A5) transporter based on dithiazole and dithiazine compounds for development of anticancer drugs
err2017-11-01
err63
errOAAI
errNapolitano, Lara; Scalise, Mariafrancesca; Koyioni, Maria; Koutentis, Panayiotis; Catto, Marco; Eberini, Ivano; Parravicini, Chiara; Palazzolo, Luca; Pisani, Leonardo; Galluccio, Michele; Console, Lara; Carotti, Angelo; Indiveri, Cesare
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Indenocinnoline derivatives as G-quadruplex binders, topoisomerase Hoc inhibitors and antiproliferative agents
err2017-05-01
err15
PREAI
errZoidis, Grigoris; Sosic, Alice; Da Ros, Silvia; Gatto, Barbara; Sissi, Claudia; Palluotto, Fausta; Carotti, Angelo; Catto, Marco
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Quinolino[3,4-b]quinoxalines and pyridazino[4,3-c]quinoline derivatives: Synthesis, inhibition of topoisomerase IIα, G-quadruplex binding and cytotoxic properties
err2016-11-01
err31
PREAI
errPalluotto, Fausta; Sosic, Alice; Pinato, Odra; Zoidis, Grigoris; Catto, Marco; Sissi, Claudia; Gatto, Barbara; Carotti, Angelo
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Exploring Basic Tail Modifications of Coumarin-Based Dual Acetylcholinesterase-Monoamine Oxidase B Inhibitors: Identification of Water-Soluble, Brain-Permeant Neuroprotective Multitarget Agents
err2016-07-07
err81
errOAAI
errPisani, Leonardo; Farina, Roberta; Catto, Marco; Iacobazzi, Rosa Maria; Nicolotti, Orazio; Cellamare, Saverio; Mangiatordi, Giuseppe Felice; Denora, Nunzio; Soto-Otero, Ramon; Siragusa, Lydia; Altomare, Cosimo Damian; Carotti, Angelo
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Searching for Multi-Targeting Neurotherapeutics against Alzheimer's: Discovery of Potent AChE-MAO B Inhibitors through the Decoration of the 2H-Chromen-2-one Structural Motif
err2016-03-17
err48
errOAAI
errPisani, Leonardo; Farina, Roberta; Soto-Otero, Ramon; Denora, Nunzio; Mangiatordi, Giuseppe Felice; Nicolotti, Orazio; Mendez-Alvarez, Estefania; Altomare, Cosimo Damiano; Catto, Marco; Carotti, Angelo
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Docking-based classification models for exploratory toxicology studies on high-quality estrogenic experimental data
err2015-10-06
err24
PREAI
errTrisciuzzi, Daniela; Alberga, Domenico; Mansouri, Kamel; Judson, Richard; Cellamare, Saverio; Catto, Marco; Carotti, Angelo; Benfenati, Emilio; Novellino, Ettore; Mangiatordi, Giuseppe Felice; Nicolotti, Orazio
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Structure-Based Design and Optimization of Multitarget-Directed 2H-Chromen-2-one Derivatives as Potent Inhibitors of Monoamine Oxidase B and Cholinesterases
err2015-07-09
err93
errOAAI
errFarina, Roberta; Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Gadaleta, Domenico; Denora, Nunzio; Soto-Otero, Ramon; Mendez-Alvarez, Estefania; Passos, Carolina S.; Muncipinto, Giovanni; Altomare, Cosimo D.; Nurisso, Alessandra; Carrupt, Pierre-Alain; Carotti, Angelo
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Multitarget-Directed Tricyclic Pyridazinones as GProtein-Coupled Receptor Ligands and Cholinesterase Inhibitors
err2015-04-29
err6
PREAI
errPau, Amedeo; Catto, Marco; Pinna, Giovanni; Frau, Simona; Murineddu, Gabriele; Asproni, Battistina; Curzu, Maria M.; Pisani, Leonardo; Leonetti, Francesco; Isabel Loza, Maria; Brea, Jose; Pinna, Gerard A.; Carotti, Angelo
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Multitarget Therapeutic Leads for Alzheimer's Disease: Quinolizidinyl Derivatives of Bi- and Tricyclic Systems as Dual Inhibitors of Cholinesterases and -Amyloid (A) Aggregation
err2015-04-29
err46
errOAAI
errTonelli, Michele; Catto, Marco; Tasso, Bruno; Novelli, Federica; Canu, Caterina; Iusco, Giovanna; Pisani, Leonardo; De Stradis, Angelo; Denora, Nunzio; Sparatore, Anna; Boido, Vito; Carotti, Angelo; Sparatore, Fabio
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Studies on the antiplatelet and antithrombotic profile of anti-inflammatory coumarin derivatives
err2015-03-25
err40
errOAAI
errKontogiorgis, Christos; Nicolotti, Orazio; Mangiatordi, Giuseppe Felice; Tognolini, Massimiliano; Karalaki, Foteini; Giorgio, Carmine; Patsilinakos, Alexandros; Carotti, Angelo; Hadjipavlou-Litina, Dimitra; Barocelli, Elisabetta
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Discovery of new 7-substituted-4-imidazolylmethyl coumarins and 4′-substituted-2-imidazolyl acetophenones open analogues as potent and selective inhibitors of steroid-11β-hydroxylase
err2015-01-01
err24
errOAAI
errStefanachi, Angela; Hanke, Nina; Pisani, Leonardo; Leonetti, Francesco; Nicolotti, Orazio; Catto, Marco; Cellamare, Saverio; Hartmann, Rolf W.; Carotti, Angelo
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In silico design of novel 2H-chromen-2-one derivatives as potent and selective MAO-B inhibitors
err2015-01-01
err60
errOAAI
errPisani, Leonardo; Farina, Roberta; Nicolotti, Orazio; Gadaleta, Domenico; Soto-Otero, Ramon; Catto, Marco; Di Braccio, Mario; Mendez-Alvarez, Estefania; Carotti, Angelo
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Computer-Aided Structure-Based Design of Multitarget Leads for Alzheimer's Disease
err2014-12-24
err46
errOAAI
errDominguez, Jose L.; Fernandez-Nieto, Fernando; Castro, Marian; Catto, Marco; Rita Paleo, M.; Porto, Silvia; Javier Sardina, F.; Brea, Jose M.; Carotti, Angelo; Carmen Villaverde, M.; Sussman, Fredy
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REACH and in silico methods: an attractive opportunity for medicinal chemists
err2014-11-01
err60
PREAI
errNicolotti, Orazio; Benfenati, Emilio; Carotti, Angelo; Gadaleta, Domenico; Gissi, Andrea; Mangiatordi, Giuseppe Felice; Novellino, Ettore
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Metabolic stability optimization and metabolite identification of 2,5-thiophene amide 17β-hydroxysteroid dehydrogenase type 2 inhibitors
err2014-11-01
err20
PREAI
errGargano, Emanuele M.; Perspicace, Enrico; Hanke, Nina; Carotti, Angelo; Marchais-Oberwinkler, Sandrine; Hartmann, Rolf W.
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First Selective Dual Inhibitors of Tau Phosphorylation and Beta-Amyloid Aggregation, Two Major Pathogenic Mechanisms in Alzheimer's Disease
err2014-09-26
err32
PREAI
errMariano, Marica; Schmitt, Christian; Miralinaghi, Parisa; Catto, Marco; Hartmann, Rolf W.; Carotti, Angelo; Engel, Matthias
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Trimethoxybenzanilide-Based P-Glycoprotein Modulators: An Interesting Case of Lipophilicity Tuning by Intramolecular Hydrogen Bonding
err2014-08-05
err24
PREAI
errTardia, Piero; Stefanachi, Angela; Niso, Mauro; Stolfa, Diana Antonella; Mangiatordi, Giuseppe Felice; Alberga, Domenico; Nicolotti, Orazio; Lattanzi, Gianluca; Carotti, Angelo; Leonetti, Francesco; Perrone, Roberto; Berardi, Francesco; Azzariti, Amalia; Colabufo, Nicola Antonio; Cellamare, Saverio
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