Not logged in Thioxanthenone-based derivatives as multitarget therapeutic leads for Alzheimer's disease Tonelli, Michele; Catto, Marco; Sabate, Raimon; Francesconi, Valeria; Laurini, Erik; Pricl, Sabrina; Pisani, Leonardo; Miniero, Daniela Valeria; Liuzzi, Grazia Maria; Gatta, Elena; Relini, Annalisa; Gavin, Rosalina; Rio, Jose Antonio Del; Sparatore, Fabio; Carotti, Angelo Share Save
17β-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer Gargano, Emanuele M.; Mohamed, Abdelrahman; Abdelsamie, Ahmed S.; Mangiatordi, Giuseppe F.; Drzewiecka, Hanna; Jagodzinski, Pawel P.; Mazzini, Arcangela; van Koppen, Chris J.; Laschke, Matthias W.; Nicolotti, Orazio; Carotti, Angelo; Marchais-Oberwinkler, Sandrine; Hartmann, Rolf W.; Frotscher, Martin Share Save
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Potent inhibitors of human LAT1 (SLC7A5) transporter based on dithiazole and dithiazine compounds for development of anticancer drugs Napolitano, Lara; Scalise, Mariafrancesca; Koyioni, Maria; Koutentis, Panayiotis; Catto, Marco; Eberini, Ivano; Parravicini, Chiara; Palazzolo, Luca; Pisani, Leonardo; Galluccio, Michele; Console, Lara; Carotti, Angelo; Indiveri, Cesare Share Save
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Quinolino[3,4-b]quinoxalines and pyridazino[4,3-c]quinoline derivatives: Synthesis, inhibition of topoisomerase IIα, G-quadruplex binding and cytotoxic properties Palluotto, Fausta; Sosic, Alice; Pinato, Odra; Zoidis, Grigoris; Catto, Marco; Sissi, Claudia; Gatto, Barbara; Carotti, Angelo Share Save
Exploring Basic Tail Modifications of Coumarin-Based Dual Acetylcholinesterase-Monoamine Oxidase B Inhibitors: Identification of Water-Soluble, Brain-Permeant Neuroprotective Multitarget Agents Pisani, Leonardo; Farina, Roberta; Catto, Marco; Iacobazzi, Rosa Maria; Nicolotti, Orazio; Cellamare, Saverio; Mangiatordi, Giuseppe Felice; Denora, Nunzio; Soto-Otero, Ramon; Siragusa, Lydia; Altomare, Cosimo Damian; Carotti, Angelo Share Save
Searching for Multi-Targeting Neurotherapeutics against Alzheimer's: Discovery of Potent AChE-MAO B Inhibitors through the Decoration of the 2H-Chromen-2-one Structural Motif Pisani, Leonardo; Farina, Roberta; Soto-Otero, Ramon; Denora, Nunzio; Mangiatordi, Giuseppe Felice; Nicolotti, Orazio; Mendez-Alvarez, Estefania; Altomare, Cosimo Damiano; Catto, Marco; Carotti, Angelo Share Save
Docking-based classification models for exploratory toxicology studies on high-quality estrogenic experimental data Trisciuzzi, Daniela; Alberga, Domenico; Mansouri, Kamel; Judson, Richard; Cellamare, Saverio; Catto, Marco; Carotti, Angelo; Benfenati, Emilio; Novellino, Ettore; Mangiatordi, Giuseppe Felice; Nicolotti, Orazio Share Save
Structure-Based Design and Optimization of Multitarget-Directed 2H-Chromen-2-one Derivatives as Potent Inhibitors of Monoamine Oxidase B and Cholinesterases Farina, Roberta; Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Gadaleta, Domenico; Denora, Nunzio; Soto-Otero, Ramon; Mendez-Alvarez, Estefania; Passos, Carolina S.; Muncipinto, Giovanni; Altomare, Cosimo D.; Nurisso, Alessandra; Carrupt, Pierre-Alain; Carotti, Angelo Share Save
Multitarget-Directed Tricyclic Pyridazinones as GProtein-Coupled Receptor Ligands and Cholinesterase Inhibitors Pau, Amedeo; Catto, Marco; Pinna, Giovanni; Frau, Simona; Murineddu, Gabriele; Asproni, Battistina; Curzu, Maria M.; Pisani, Leonardo; Leonetti, Francesco; Isabel Loza, Maria; Brea, Jose; Pinna, Gerard A.; Carotti, Angelo Share Save
Multitarget Therapeutic Leads for Alzheimer's Disease: Quinolizidinyl Derivatives of Bi- and Tricyclic Systems as Dual Inhibitors of Cholinesterases and -Amyloid (A) Aggregation Tonelli, Michele; Catto, Marco; Tasso, Bruno; Novelli, Federica; Canu, Caterina; Iusco, Giovanna; Pisani, Leonardo; De Stradis, Angelo; Denora, Nunzio; Sparatore, Anna; Boido, Vito; Carotti, Angelo; Sparatore, Fabio Share Save
Studies on the antiplatelet and antithrombotic profile of anti-inflammatory coumarin derivatives Kontogiorgis, Christos; Nicolotti, Orazio; Mangiatordi, Giuseppe Felice; Tognolini, Massimiliano; Karalaki, Foteini; Giorgio, Carmine; Patsilinakos, Alexandros; Carotti, Angelo; Hadjipavlou-Litina, Dimitra; Barocelli, Elisabetta Share Save
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Computer-Aided Structure-Based Design of Multitarget Leads for Alzheimer's Disease Dominguez, Jose L.; Fernandez-Nieto, Fernando; Castro, Marian; Catto, Marco; Rita Paleo, M.; Porto, Silvia; Javier Sardina, F.; Brea, Jose M.; Carotti, Angelo; Carmen Villaverde, M.; Sussman, Fredy Share Save
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Trimethoxybenzanilide-Based P-Glycoprotein Modulators: An Interesting Case of Lipophilicity Tuning by Intramolecular Hydrogen Bonding Tardia, Piero; Stefanachi, Angela; Niso, Mauro; Stolfa, Diana Antonella; Mangiatordi, Giuseppe Felice; Alberga, Domenico; Nicolotti, Orazio; Lattanzi, Gianluca; Carotti, Angelo; Leonetti, Francesco; Perrone, Roberto; Berardi, Francesco; Azzariti, Amalia; Colabufo, Nicola Antonio; Cellamare, Saverio Share Save