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Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T. Share Save
Green Synthesis of Sulfonamide Derivatives as Human Carbonic Anhydrase Isoforms I, II, IX, XII Inhibitors and Antioxidants: Comprehensive Insights From Biological Evaluation and In-Depth In Silico Analysis Mishra, K. M. Abha; Kumari, Nutan; Carta, Fabrizio; Renzi, Gioele; Singh, Harshdeep; Supuran, Claudiu T.; Sethi, Kalyan K. Share Save
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Unraveling the Potential of Amino-, Acylamino-, and Ureido-Substituted 3H-1,2-Benzoxaphosphepine 2-Oxides toward Nanomolar Inhibitors of Tumor-Associated Carbonic Anhydrases IX and XII Balasova, A; Pustenko, A; Angeli, A; Andreucci, E; Biagioni, A; Nocentini, A; Carta, F; Supuran, CT; Zalubovskis, R Share Save
Discovery of Trypanosoma cruzi Carbonic Anhydrase Inhibitors by a Combination of Ligand- and Structure-Based Virtual Screening Gori, Denis N. Prada; Barrionuevo, Emilia M.; Alberca, Lucas N.; Sbaraglini, Maria L.; Llanos, Manuel A.; Giovannuzzi, Simone; Carta, Fabrizio; Marchetto, Matias I.; Supuran, Claudiu T.; Soto, Catalina D. Alba; Gavernet, Luciana; Talevi, Alan Share Save
Discover the Power of Lithospermic Acid as Human Carbonic Anhydrase VA and Pancreatic Lipase Inhibitor Through In Silico and In Vitro Studies Citriniti, Emanuele Liborio; Rocca, Roberta; Costa, Giosue; Sciacca, Claudia; Cardullo, Nunzio; Muccilli, Vera; Karioti, Anastasia; Carta, Fabrizio; Supuran, Claudiu T.; Alcaro, Stefano; Ortuso, Francesco Share Save
In Vitro CO-Releasing and Antioxidant Properties of Sulfonamide-Based CAI-CORMs in a H2O2-Stimulated Human Achilles Tendon-Derived Cell Model Berrino, Emanuela; Guglielmi, Paolo; Carta, Fabrizio; Carradori, Simone; Campestre, Cristina; Angeli, Andrea; Arrighi, Francesca; Pontecorvi, Virginia; Chimenti, Paola; Secci, Daniela; Supuran, Claudiu T.; Gallorini, Marialucia Share Save
Design, Synthesis, and In Vitro Evaluation of Aromatic Sulfonamides as Human Carbonic Anhydrase I, II, IX, and XII Inhibitors and Their Antioxidant Activity Mishra, K. M. Abha; Kumari, Nutan; Carta, Fabrizio; Renzi, Gioele; Supuran, Claudiu T.; Sethi, Kalyan K. Share Save
X-ray crystallographic and kinetic studies of biguanide containing aryl sulfonamides as carbonic anhydrase inhibitors Baroni, Chiara; Bozdag, Murat; Renzi, Gioele; De Luca, Viviana; Capasso, Clemente; Bazzicalupi, Carla; Selleri, Silvia; Ferraroni, Marta; Carta, Fabrizio; Supuran, Claudiu T. Share Save
Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms Kilbile, Jaydeo T.; Sapkal, Suryakant B.; Renzi, Gioele; D'Agostino, Ilaria; Boudjelal, Mohamed; Tamboli, Yasinalli; Cutarella, Luigi; Mori, Mattia; Sgambellone, Silvia; Villano, Serafina; Marri, Silvia; Lucarini, Laura; Carradori, Simone; Carta, Fabrizio; Supuran, Claudiu T. Share Save
Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study Marinacci, Beatrice; D'Agostino, Ilaria; Angeli, Andrea; Carradori, Simone; Melfi, Francesco; Grande, Rossella; Corsiani, Micol; Ferraroni, Marta; Agamennone, Mariangela; Tondo, Anna Rita; Zara, Susi; Puca, Valentina; Pellegrini, Benedetta; Vagaggini, Chiara; Dreassi, Elena; Patrauchan, Marianna A.; Capasso, Clemente; Nicolotti, Orazio; Carta, Fabrizio; Supuran, Claudiu T. Share Save
Superacid-Synthesized Fluorinated Diamines Act as Selective hCA IV Inhibitors Berrino, Emanuela; Michelet, Bastien; Vitse, Kassandra; Nocentini, Alessio; Bartolucci, Gianluca; Martin-Mingot, Agnes; Gratteri, Paola; Carta, Fabrizio; Supuran, Claudiu T.; Thibaudeau, Sebastien Share Save
Lasamide, a Potent Human Carbonic Anhydrase Inhibitor from the Market: Inhibition Profiling and Crystallographic Studies Baroni, Chiara; D'Agostino, Ilaria; Renzi, Gioele; Kilbile, Jaydeo T.; Tamboli, Yasinalli; Ferraroni, Marta; Carradori, Simone; Capasso, Clemente; Carta, Fabrizio; Supuran, Claudiu T. Share Save
2-Substituted-4,7-dihydro-4-ethylpyrazolo[1,5- a ]pyrimidin-7-ones alleviate LPS-induced inflammation by modulating cell metabolism via CD73 upon macrophage polarization Ricci, Alessia; Zara, Susi; Carta, Fabrizio; Di Valerio, Valentina; Sancilio, Silvia; Cataldi, Amelia; Selleri, Silvia; Supuran, Claudiu T.; Carradori, Simone; Gallorini, Marialucia Share Save