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Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino [4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults Samarelli, Francesco; Purgatorio, Rosa; Lopopolo, Gianfranco; Deruvo, Caterina; Catto, Marco; Andresini, Michael; Carrieri, Antonio; Nicolotti, Orazio; De Palma, Annalisa; Miniero, Daniela Valeria; de Candia, Modesto; Altomare, Cosimo D. Share Save
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Microwave-Assisted Extraction of Bioactive Compounds from Lentil Wastes: Antioxidant Activity Evaluation and Metabolomic Characterization Cavalluzzi, Maria Maddalena; Lamonaca, Antonella; Rotondo, Natalie Paola; Miniero, Daniela Valeria; Muraglia, Marilena; Gabriele, Paola; Corbo, Filomena; De Palma, Annalisa; Budriesi, Roberta; De Angelis, Elisabetta; Monaci, Linda; Lentini, Giovanni Share Save
Densely Functionalized 2-Methylideneazetidines: Evaluation as Antibacterials Petrillo, Giovanni; Tavani, Cinzia; Bianchi, Lara; Benzi, Alice; Cavalluzzi, Maria Maddalena; Salvagno, Lara; Quintieri, Laura; De Palma, Annalisa; Caputo, Leonardo; Rosato, Antonio; Lentini, Giovanni Share Save
Synthesis and Evaluation of Voltage-Gated Sodium Channel Blocking Pyrroline Derivatives Endowed with Both Antiarrhythmic and Antioxidant Activities Carocci, Alessia; Roselli, Mariagrazia; Budriesi, Roberta; Micucci, Matteo; Desaphy, Jean-Francois; Altamura, Concetta; Cavalluzzi, Maria Maddalena; Toma, Maddalena; Passeri, Giovanna Ilaria; Milani, Gualtiero; Lovece, Angelo; Catalano, Alessia; Bruno, Claudio; De Palma, Annalisa; Corbo, Filomena; Franchini, Carlo; Habtemariam, Solomon; Lentini, Giovanni Share Save
Scouting around 1,2,3,4-Tetrahydrochromeno[3,2-c]pyridin-10-ones for Single- and Multitarget Ligands Directed towards Relevant Alzheimer's Targets Purgatorio, Rosa; Kulikova, Larisa N.; Pisani, Leonardo; Catto, Marco; de Candia, Modesto; Carrieri, Antonio; Cellamare, Saverio; De Palma, Annalisa; Beloglazkin, Andrey A.; Reza Raesi, Ghulam; Voskressensky, Leonid G.; Altomare, Cosimo D. Share Save
Chiral Separation, X-ray Structure, and Biological Evaluation of a Potent and Reversible Dual Binding Site AChE Inhibitor Catto, Marco; Pisani, Leonardo; de la Mora, Eugenio; Belviso, Benny Danilo; Mangiatordi, Giuseppe Felice; Pinto, Andrea; De Palma, Annalisa; Denora, Nunzio; Caliandro, Rocco; Colletier, Jacques-Philippe; Silman, Israel; Nicolotti, Orazio; Altomare, Cosimo Damiano Share Save
Investigating 1,2,3,4,5,6-hexahydroazepino[4,3-b]indole as scaffold of butyrylcholinesterase-selective inhibitors with additional neuroprotective activities for Alzheimer's disease Purgatorio, Rosa; de Candia, Modesto; Catto, Marco; Carrieri, Antonio; Pisani, Leonardo; De Palma, Annalisa; Toma, Maddalena; Ivanova, Olga A.; Voskressensky, Leonid G.; Altomare, Cosimo D. Share Save
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Mannich base approach to 5-methoxyisatin 3-(4-isopropylphenyl) hydrazone: A water-soluble prodrug for a multitarget inhibition of cholinesterases, beta-amyloid fibrillization and oligomer-induced cytotoxicity Pisani, Leonardo; De Palma, Annalisa; Giangregorio, Nicola; Miniero, Daniela V.; Pesce, Paolo; Nicolotti, Orazio; Campagna, Francesco; Altomare, Cosimo D.; Catto, Marco Share Save
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Synthesis, antiarrhythmic activity, and toxicological evaluation of mexiletine analogues Roselli, Mariagrazia; Carocci, Alessia; Budriesi, Roberta; Micucci, Matteo; Toma, Maddalena; Mannelli, Lorenzo Di Cesare; Lovece, Angelo; Catalano, Alessia; Cavalluzzi, Maria Maddalena; Bruno, Claudio; De Palma, Annalisa; Contino, Marialessandra; Perrone, Maria Grazia; Colabufo, Nicola Antonio; Chiarini, Alberto; Franchini, Carlo; Ghelardini, Carla; Habtemariam, Solomon; Lentini, Giovanni Share Save
N-(Phenoxyalkyl)amides as MT1 and MT2 ligands: Antioxidant properties and inhibition of Ca2+/CaM-dependent kinase II Carocci, Alessia; Catalano, Alessia; Bruno, Claudio; Lovece, Angelo; Roselli, Maria Grazia; Cavalluzzi, Maria Maddalena; De Santis, Francesco; De Palma, Annalisa; Rusciano, Maria Rosaria; Illario, Maddalena; Franchini, Carlo; Lentini, Giovanni Share Save
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Synthesis and Toxicopharmacological Evaluation of m-Hydroxymexiletine, the First Metabolite of Mexiletine More Potent Than the Parent Compound on Voltage-Gated Sodium Channels Catalano, Alessia; Desaphy, Jean-Francois; Lentini, Giovanni; Carocci, Alessia; Di Mola, Antonia; Bruno, Claudio; Carbonara, Roberta; De Palma, Annalisa; Budriesi, Roberta; Ghelardini, Carla; Perrone, Maria Grazia; Colabufo, Nicola Antonio; Camerino, Diana Conte; Franchini, Carlo Share Save
New N-(phenoxydecyl) phthalimide derivatives displaying potent inhibition activity towards α-glucosidase Pascale, Rossana; Carocci, Alessia; Catalano, Alessia; Lentini, Giovanni; Spagnoletta, Anna; Cavalluzzi, Maria Maddalena; De Santis, Francesco; De Palma, Annalisa; Scalera, Vito; Franchini, Carlo Share Save