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Annalisa De Palma

University of Bari Aldo Moro

18H-index
47Paper Count
1.0KCitation Count
Published Papers 21
Publication Date
Exploring Pyrazolidinone and Pyrazolidinedione Scaffolds for Alzheimer's Therapy: Multitarget COX-2 Inhibitors with Anti-Amyloid β; Anti-Tau; Antioxidant; and Neuroprotective Activities
err2025-11-10
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PREAI
errMichael Emad; Reham Waheed; Zeinab Mostafa; Sarah S Darwish; Rosa Purgatorio; Daniela V Miniero; Annalisa De Palma; Tzu-Peng Cheng; Yu-Cheng Chen; Moustafa Gabr; Ahmed M El Kerdawy; Marco Catto; Ashraf H. Abadi; Tsong-Long Hwang; Mohammad Abdel-Halim
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Revisiting COX-2 Inhibitors for Alzheimer's Disease as Multitargeted Ligands: Development of 4-Hydrazono-Pyrazolidinediones with Tuned COX Selectivity Profile and Improved Cellular Potency
err2025-10-13
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PREAI
errReham Waheed; Zeinab Moustafa; Michael Emad; Sarah S. Darwish; Rosa Purgatorio; Daniela Valeria Miniero; Annalisa De Palma; Tzu-Peng Cheng; Ting-Yu Wang; Yu-Cheng Chen; Ahmed M. El Kerdawy; Moustafa T. Gabr; Marco Catto; Ashraf H. Abadi; Tsong-Long Hwang; Mohammad Abdel-Halim
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Modulatory Effect of Nicotinamide Adenine Dinucleotide Phosphate (NADPH) on the 2-Oxoglutarate Mitochondrial Carrier
err2024-10-31
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errOAAI
errSpagnoletta, Anna; Miniero, Daniela Valeria; Gambacorta, Nicola; Oppedisano, Francesca; De Grassi, Anna; Nicolotti, Orazio; Pierri, Ciro Leonardo; De Palma, Annalisa
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Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino [4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults
err2024-04-01
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errSamarelli, Francesco; Purgatorio, Rosa; Lopopolo, Gianfranco; Deruvo, Caterina; Catto, Marco; Andresini, Michael; Carrieri, Antonio; Nicolotti, Orazio; De Palma, Annalisa; Miniero, Daniela Valeria; de Candia, Modesto; Altomare, Cosimo D.
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New Insights Regarding Hemin Inhibition of the Purified Rat Brain 2-Oxoglutarate Carrier and Relationships with Mitochondrial Dysfunction
err2022-12-19
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errMiniero, Daniela Valeria; Gambacorta, Nicola; Spagnoletta, Anna; Tragni, Vincenzo; Loizzo, Stefano; Nicolotti, Orazio; Pierri, Ciro Leonardo; De Palma, Annalisa
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Microwave-Assisted Extraction of Bioactive Compounds from Lentil Wastes: Antioxidant Activity Evaluation and Metabolomic Characterization
err2022-11-02
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errCavalluzzi, Maria Maddalena; Lamonaca, Antonella; Rotondo, Natalie Paola; Miniero, Daniela Valeria; Muraglia, Marilena; Gabriele, Paola; Corbo, Filomena; De Palma, Annalisa; Budriesi, Roberta; De Angelis, Elisabetta; Monaci, Linda; Lentini, Giovanni
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Densely Functionalized 2-Methylideneazetidines: Evaluation as Antibacterials
err2021-06-25
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errPetrillo, Giovanni; Tavani, Cinzia; Bianchi, Lara; Benzi, Alice; Cavalluzzi, Maria Maddalena; Salvagno, Lara; Quintieri, Laura; De Palma, Annalisa; Caputo, Leonardo; Rosato, Antonio; Lentini, Giovanni
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Synthesis and Evaluation of Voltage-Gated Sodium Channel Blocking Pyrroline Derivatives Endowed with Both Antiarrhythmic and Antioxidant Activities
err2020-10-28
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PREAI
errCarocci, Alessia; Roselli, Mariagrazia; Budriesi, Roberta; Micucci, Matteo; Desaphy, Jean-Francois; Altamura, Concetta; Cavalluzzi, Maria Maddalena; Toma, Maddalena; Passeri, Giovanna Ilaria; Milani, Gualtiero; Lovece, Angelo; Catalano, Alessia; Bruno, Claudio; De Palma, Annalisa; Corbo, Filomena; Franchini, Carlo; Habtemariam, Solomon; Lentini, Giovanni
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Scouting around 1,2,3,4-Tetrahydrochromeno[3,2-c]pyridin-10-ones for Single- and Multitarget Ligands Directed towards Relevant Alzheimer's Targets
err2020-09-04
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PREAI
errPurgatorio, Rosa; Kulikova, Larisa N.; Pisani, Leonardo; Catto, Marco; de Candia, Modesto; Carrieri, Antonio; Cellamare, Saverio; De Palma, Annalisa; Beloglazkin, Andrey A.; Reza Raesi, Ghulam; Voskressensky, Leonid G.; Altomare, Cosimo D.
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Chiral Separation, X-ray Structure, and Biological Evaluation of a Potent and Reversible Dual Binding Site AChE Inhibitor
err2020-02-07
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errCatto, Marco; Pisani, Leonardo; de la Mora, Eugenio; Belviso, Benny Danilo; Mangiatordi, Giuseppe Felice; Pinto, Andrea; De Palma, Annalisa; Denora, Nunzio; Caliandro, Rocco; Colletier, Jacques-Philippe; Silman, Israel; Nicolotti, Orazio; Altomare, Cosimo Damiano
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Investigating 1,2,3,4,5,6-hexahydroazepino[4,3-b]indole as scaffold of butyrylcholinesterase-selective inhibitors with additional neuroprotective activities for Alzheimer's disease
err2019-09-01
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errPurgatorio, Rosa; de Candia, Modesto; Catto, Marco; Carrieri, Antonio; Pisani, Leonardo; De Palma, Annalisa; Toma, Maddalena; Ivanova, Olga A.; Voskressensky, Leonid G.; Altomare, Cosimo D.
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Insights into Structure-Activity Relationships of 3-Arylhydrazonoindolin-2-One Derivatives for Their Multitarget Activity on β-Amyloid Aggregation and Neurotoxicity
err2018-06-26
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errPurgatorio, Rosa; de Candia, Modesto; De Palma, Annalisa; De Santis, Francesco; Pisani, Leonardo; Campagna, Francesco; Cellamare, Saverio; Altomare, Cosimo Damiano; Catto, Marco
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Mannich base approach to 5-methoxyisatin 3-(4-isopropylphenyl) hydrazone: A water-soluble prodrug for a multitarget inhibition of cholinesterases, beta-amyloid fibrillization and oligomer-induced cytotoxicity
err2017-11-01
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errPisani, Leonardo; De Palma, Annalisa; Giangregorio, Nicola; Miniero, Daniela V.; Pesce, Paolo; Nicolotti, Orazio; Campagna, Francesco; Altomare, Cosimo D.; Catto, Marco
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Nitric oxide inhibits the mitochondrial carnitine/acylcarnitine carrier through reversible S-nitrosylation of cysteine 136
err2017-07-01
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errTonazzi, Annamaria; Giangregorio, Nicola; Console, Lara; De Palma, Annalisa; Indiveri, Cesare
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Discovery of Potent Dual Binding Site Acetylcholinesterase Inhibitors via Homo- and Heterodimerization of Coumarin-Based Moieties
err2017-06-29
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errPisani, Leonardo; Catto, Marco; De Palma, Annalisa; Farina, Roberta; Cellamare, Saverio; Altomare, Cosimo D.
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Synthesis, antiarrhythmic activity, and toxicological evaluation of mexiletine analogues
err2016-10-01
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errRoselli, Mariagrazia; Carocci, Alessia; Budriesi, Roberta; Micucci, Matteo; Toma, Maddalena; Mannelli, Lorenzo Di Cesare; Lovece, Angelo; Catalano, Alessia; Cavalluzzi, Maria Maddalena; Bruno, Claudio; De Palma, Annalisa; Contino, Marialessandra; Perrone, Maria Grazia; Colabufo, Nicola Antonio; Chiarini, Alberto; Franchini, Carlo; Ghelardini, Carla; Habtemariam, Solomon; Lentini, Giovanni
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N-(Phenoxyalkyl)amides as MT1 and MT2 ligands: Antioxidant properties and inhibition of Ca2+/CaM-dependent kinase II
err2013-02-01
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PREAI
errCarocci, Alessia; Catalano, Alessia; Bruno, Claudio; Lovece, Angelo; Roselli, Maria Grazia; Cavalluzzi, Maria Maddalena; De Santis, Francesco; De Palma, Annalisa; Rusciano, Maria Rosaria; Illario, Maddalena; Franchini, Carlo; Lentini, Giovanni
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Decreased expression of the Augmenter of Liver Regeneration results in increased apoptosis and oxidative damage in human-derived glioma cells
err2012-04-05
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errOAAI
errPolimeno, L.; Pesetti, B.; De Santis, F.; Resta, L.; Rossi, R.; De Palma, A.; Girardi, B.; Amoruso, A.; Francavilla, A.
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Synthesis and Toxicopharmacological Evaluation of m-Hydroxymexiletine, the First Metabolite of Mexiletine More Potent Than the Parent Compound on Voltage-Gated Sodium Channels
err2012-01-31
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PREAI
errCatalano, Alessia; Desaphy, Jean-Francois; Lentini, Giovanni; Carocci, Alessia; Di Mola, Antonia; Bruno, Claudio; Carbonara, Roberta; De Palma, Annalisa; Budriesi, Roberta; Ghelardini, Carla; Perrone, Maria Grazia; Colabufo, Nicola Antonio; Camerino, Diana Conte; Franchini, Carlo
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New N-(phenoxydecyl) phthalimide derivatives displaying potent inhibition activity towards α-glucosidase
err2010-08-01
err48
PREAI
errPascale, Rossana; Carocci, Alessia; Catalano, Alessia; Lentini, Giovanni; Spagnoletta, Anna; Cavalluzzi, Maria Maddalena; De Santis, Francesco; De Palma, Annalisa; Scalera, Vito; Franchini, Carlo
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