未登录Identification and Biological Evaluation of (4H-Thieno[3,2-b]indol-3-yl)methanol as a Tumoricidal Scaffold for an Antineoplastic Agent
Zhuang, Shi-Hong; Chang, Yi-Han; Huynh, Hoang-Thuc; Hung, Hsin-Yi; Huang, Zih-Ting; Juang, Shin-Hun; Kuo, Sheng-Chu; Kuo, Ching-Chuan; Hsieh, Min-Tsang
分享
收藏
分享
收藏
分享
收藏Cytotoxicity-guided isolation of elatostemanosides I-VI from Elatostema tenuicaudatum W. T. Wang and their cytotoxic activities基于细胞毒性的Elatostema tenuicaudatum W. T. Wang中Elatostemanosides I-VI的分离及其细胞毒性活性
Huynh, Quoc-Dung Tran; Phan, Thuy-Tien Thi; Liu, Ta-Wei; Duong, Truc-Ly Thi; Hsu, Su-Jung; Kuo, Ching-Chuan; Chu, Man-Hsiu; Wang, Yun-Han; Nguyen, Thanh-Vu; Shen, Yao-An; Fan, Yu-Jui; Nguyen, Dang-Khoa; Vo, Thanh-Hoa
分享
收藏Development of Potent and Selective Inhibitors of Methylenetetrahydrofolate Dehydrogenase 2 for Targeting Acute Myeloid Leukemia: SAR, Structural Insights, and Biological Characterization
Chang, Hsin-Huei; Lee, Lung-Chun; Hsu, Tsu; Peng, Yi-Hui; Huang, Chih-Hsiang; Yeh, Teng-Kuang; Lu, Cheng-Tai; Huang, Zih-Ting; Hsueh, Ching-Cheng; Kung, Fang-Chun; Lin, Li-Mei; Huang, Yu-Chen; Wang, Yi-Hsin; Li, Li-Hsuan; Tang, Ya-Chu; Chang, Ling; Hsieh, Chih-Chien; Jiaang, Weir-Torn; Kuo, Ching-Chuan; Wu, Su-Ying
分享
收藏
分享
收藏Lysosomal-targeted doxorubicin delivery using RBC-derived vesicles to overcome drug-resistant cancer through mitochondrial-dependent cell death
Lin, Chih-Peng; Wu, Shu-Hui; Lin, Tzu-Yin; Chu, Chia-Hui; Lo, Leu-Wei; Kuo, Ching-Chuan; Chang, Jang-Yang; Hsu, Szu-Chun; Ko, Bor-Sheng; Yao, Ming; Hsiao, Jong-Kai; Wang, Shih-Wei; Huang, Dong-Ming
分享
收藏Discovery and development of a novel N-(3-bromophenyl)- {[(phenylcarbamoyl)amino]methyl}-N-hydroxythiophene-2-carboximidamide indoleamine 2,3-dioxygenase inhibitor using knowledge-based drug design使用基于知识的药物设计发现和开发新型N-(3-溴苯基)- {[(苯基氨基甲酰基) 氨基] 甲基}-N-hydroxythiophene-2-carboximidamide吲哚胺2,3-双加氧酶抑制剂
Yeh, Teng-Kuang; Song, Jen-Shin; Chang, Po-Wei; Yu, Jin-Chen; Chang, Chia-Hwa; Liao, Fang-Yu; Tien, Ya-Wen; Kuppusamy, Ramajayam; Li, An-Siou; Chen, Chi-Han; Chen, Chieh-Wen; Lin, Li-Mei; Chang, Hsin-Huei; Huang, Chih-Hsiang; Yao, Jau-Ying; Wu, Mine-Hsine; Peng, Yi-Hui; Hsueh, Ching-Cheng; Hsiao, Wen-Chi; Chen, Pei-Husan; Lin, Chin-Yu; Hsieh, Su-Huei; Shih, Chuan; Hung, Ming-Shiu; Wu, Su-Ying; Kuo, Ching-Chuan; Ueng, Shau-Hua
分享
收藏
分享
收藏Type-3 Hyaluronan Synthase Attenuates Tumor Cells Invasion in Human Mammary Parenchymal Tissues
Lee, Wen-Jui; Tu, Shih-Hsin; Cheng, Tzu-Chun; Lin, Juo-Han; Sheu, Ming-Thau; Kuo, Ching-Chuan; Changou, Chun A.; Wu, Chih-Hsiung; Chang, Hui-Wen; Chang, Hang-Lung; Chen, Li-Ching; Ho, Yuan-Soon
分享
收藏Xanthine Derivatives Reveal an Allosteric Binding Site in Methylenetetrahydrofolate Dehydrogenase 2 (MTHFD2)
Lee, Lung-Chun; Peng, Yi-Hui; Chang, Hsin-Huei; Hsu, Tsu; Lu, Cheng-Tai; Huang, Chih-Hsiang; Hsueh, Ching-Cheng; Kung, Fang-Chun; Kuo, Ching-Chuan; Jiaang, Weir-Torn; Wu, Su-Ying
分享
收藏c-MYC-directed NRF2 drives malignant progression of head and neck cancer via glucose-6-phosphate dehydrogenase and transketolase activation
Tang, Ya-Chu; Hsiao, Jenn-Ren; Jiang, Shih-Sheng; Chang, Jang-Yang; Chu, Pei-Yi; Liu, Ko-Jiunn; Fang, Hsun-Lang; Lin, Li-Mei; Chen, Huang-Hui; Huang, Yen-Wen; Chen, Yu-Tsen; Tsai, Fang-Yu; Lin, Su-Fang; Chuang, Yung-Jen; Kuo, Ching-Chuan
分享
收藏Unique Sulfur-Aromatic Interactions Contribute to the Binding of Potent Imidazothiazole Indoleamine 2,3-Dioxygenase Inhibitors (vol 63, pg 1642, 2020)
Peng, Yi-Hui; Liao, Fang-Yu; Tseng, Chen-Tso; Kuppusamy, Ramajayam; Li, An-Siou; Chen, Chi-Han; Fan, Yu-Shiou; Wang, Sing-Yi; Wu, Mine-Hsine; Hsueh, Ching-Cheng; Chang, Jia-Yu; Lee, Lung-Chun; Shih, Chuan; Shia, Kak-Shan; Yeh, Teng-Kuang; Hung, Ming-Shiu; Kuo, Ching-Chuan; Song, Jen-Shin; Wu, Su-Ying; Ueng, Shau-Hua
分享
收藏
分享
收藏Unique Sulfur-Aromatic Interactions Contribute to the Binding of Potent Imidazothiazole Indoleamine 2,3-Dioxygenase Inhibitors
Peng, Yi-Hui; Liao, Fang-Yu; Tseng, Chen-Tso; Kuppusamy, Ramajayam; Li, An-Siou; Chen, Chi-Han; Fan, Yu-Shiou; Wang, Sing-Yi; Wu, Mine-Hsine; Hsueh, Ching-Cheng; Chang, Jia-Yu; Lee, Lung-Chun; Shih, Chuan; Shia, Kak-Shan; Yeh, Teng-Kuang; Hung, Ming-Shiu; Kuo, Ching-Chuan; Song, Jen-Shin; Wu, Su-Ying; Ueng, Shau-Hua
分享
收藏Identification of a Multitargeted Tyrosine Kinase Inhibitor for the Treatment of Gastrointestinal Stromal Tumors and Acute Myeloid Leukemia
Lin, Wen-Hsing; Wu, Su-Ying; Yeh, Teng-Kuang; Chen, Chiung-Tong; Song, Jen-Shin; Shiao, Hui-Yi; Kuo, Ching-Chuan; Hsu, Tsu; Lu, Cheng-Tai; Wang, Pei-Chen; Wu, Tsung-Sheng; Peng, Yi-Hui; Lin, Hui-You; Chen, Ching-Ping; Weng, Ya-Ling; Kung, Fang-Chun; Wu, Mine-Hsine; Su, Yu-Chieh; Huang, Kuo-Wei; Chou, Ling-Hui; Hsueh, Ching-Cheng; Yen, Kuei-Jung; Kuo, Po-Chu; Huang, Chen-Lung; Chen, Li-Tzong; Shih, Chuan; Tsai, Hui-Jen; Jiaang, Weir-Torn
分享
收藏Use of integrated genomic analyses in patient-derived tumor model to discover new clinical indications for the multikinase inhibitor drug candidate, DBPR216
Kuo, Ching-Chuan; Jiaang, Weir-Torn; Ou, Jing-Jim; Chen, Chiung-Tong; Hsu, Shu-Ching; Shih, Chuan; Lin, Li-Mei; Sun, Manwu; Wang, Yi-Hsin; Huang, Zih-Ting; Chang, Jang-Yang; Ueng, Shau-Hua
分享
收藏
分享
收藏
分享
收藏
分享
收藏