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徐云根 封面图

徐云根 (Yungen Xu)

china pharmaceutical university

34H指数
191论文数
3.5K被引数
收录论文 96
发表时间
Discovery of Highly Potent Phthalazinone Derivatives as PARP14 Inhibitors: From Structure-Based Virtual Screening to In Vivo Pharmacodynamic Activity基于结构的虚拟筛选发现的高效邻苯二甲氢吲哚酮衍生物作为PARP14抑制剂:从虚拟筛选到体内药效学研究
err2026-04-20
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PREAI
errShiqi Wu; Kaiyuan Cong; Jing Liu; Le Qu; Xiaorong Zeng; Xiangying Kong; Ziyue Li; Shaoxue Lou; Ping Wei; Li Shao; Hongfeng Gu; Yan Zhao; Qinlong Xu; Zhaoxing Chu; Guangwei He; Qihua Zhu; Yungen Xu; Yi Zou
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Identification of an Orally Bioavailable Quinoline-Based Small-Molecule Tumor Necrosis Factor α (TNF-α) Inhibitor Featuring a Spirocyclic Scaffold一种具有螺环骨架、口服生物利用度的喹啉基小分子肿瘤坏死因子α(TNF-α)抑制剂的鉴定
err2026-03-31
err0
PREAI
errZeren Sun; Wenbin Zhang; Wanyong He; Jie Xu; Boning Wang; Joshua M. He; Yuchen Zhang; Pu Chen; Yao Luo; Jia Gu; Hongfeng Gu; Ping Wei; Yanan Sun; Chunxiang Yin; Hanxi Xing; Yannan Luo; Jing-jing Zhang; Qihua Zhu; Yi Zou; Yungen Xu
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Discovery of Novel Orally Bioavailable Polθ Inhibitors with Arylalkyne Scaffolds for Targeting HR-Deficient Cancers
err2026-01-29
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PREAI
errJinyang Zhang; Xiaomeng Sun; Qichen Zhou; Yingying Wei; Biao Chen; Junhui Jiao; Yu Du; Shepherd Wufoyrwoth; Haoze Chi; Yi Yang; Ping Wei; Yungen Xu; Yi Zou; Qihua Zhu
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Discovery of a spirocyclic influenza RNA-dependent RNA polymerase inhibitor发现一种螺环状流感RNA依赖性RNA聚合酶抑制剂
err2025-10-17
err0
PREAI
errJianxun He; Zhaoxing Chu; Qinlong Xu; Yi Zou; Gaofeng Lin; Jiajia Mo; Li Shao; Yan Zhao; Jiaming Li; Wenfeng Ye; Tao Fang; Qihua Zhu; Guangwei He; Yungen Xu
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Discovery of Orally Potent Small-Molecule CD73 Inhibitor for Cancer Immunotherapy发现一种口服有效的用于癌症免疫治疗的小分子CD73抑制剂
err2025-05-23
err0
PREAI
errCen, Lifang; Ren, Weijie; Yu, Jiajie; Cheng, Ming; Kong, Xiangying; Yan, Wenxin; Wang, Luhua; Li, Xinyue; Liu, Jing; Wang, Zhen; Wu, Shiqi; Sun, Xiaomeng; Wei, Ping; Gu, Hongfeng; Zhu, Qihua; Zou, Yi; Xu, Yungen
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Discovery of novel JAK3 inhibitors for the treatment of atopic dermatitis发现新型JAK3抑制剂用于治疗特应性皮炎
err2025-04-24
err0
PREAI
errRen, Weijie; Cen, Lifang; Li, Xinyue; Yu, Jiajie; Wu, Shiqi; Liu, Jing; Wang, Luhua; Kong, Xiangying; Zou, Yi; Xu, Yungen
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Parps in immune response: Potential targets for cancer immunotherapy
err2025-04-01
err1
PREAI
errWang, Shuping; Huang, Jingling; Zeng, Tingyu; Chen, Yali; Xu, Yungen; Zhang, Bangzhi
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Design, synthesis, and antitumor evaluation of triazolopyridine derivatives as novel inhibitors for BRD4
err2025-03-01
err0
PREAI
errLiu, Jing-Ying; Zhang, Hong-En; Wang, Cheng; Zhang, Ping-Fan; Xu, Yun-Gen; Shi, Lei; Sun, Li-Ping
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New TIPARP inhibitor rescues mitochondrial function and brain injury in ischemic stroke
err2024-12-01
err0
errOAAI
errCai, Yang; Gu, Hongfeng; Li, Lu; Liu, Xue; Bai, Ying; Shen, Ling; Han, Bing; Xu, Yungen; Yao, Honghong
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Discovery of cyanoguanidine derivatives as biased μ-opioid receptor agonists
err2024-11-01
err1
PREAI
errZhu, Liang-han; Mao, Hui-huan; He, Mingchao; Cui, Zhi-ying; Zhu, Qi-hua; Gu, Hong-feng; Xu, Yun-gen
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Discovery of novel EGFR-PROTACs capable of degradation of multiple EGFR-mutated proteins能够降解多种EGFR突变蛋白的新型egfr-protacs的发现
err2024-06-01
err8
PREAI
errDu, Yu; Shi, Shi; Shu, Chen; He, Yezi; Xu, Wangyang; Wu, Daochen; Tian, Yushu; Kong, Mingyang; He, Jiahuan; Xie, Wenhui; Qiu, Yijia; Xu, Yungen; Zou, Yi; Zhu, Qihua
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Rational Design of PARP1/c-Met Dual Inhibitors for Overcoming PARP1 Inhibitor Resistance Induced by c-Met Overexpression
err2024-03-13
err5
PREAI
errSun, Zeren; Li, Lanjie; Zhai, Bingxin; Hu, Mengxuan; Huang, Lei; Huang, Shihui; Ye, Liu; Kong, Xiangying; Xu, Jie; Bai, Jie; Yan, Jingjie; Zhou, Qichen; Hu, Zheqi; Zhang, Yuchen; Jiang, Yuhan; Zhang, Yan; Qiao, Zhou; Zou, Yi; Xu, Yungen; Zhu, Qihua
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Discovery of the first ataxia telangiectasia and Rad3-related (ATR) degraders for cancer treatment
err2024-03-01
err1
PREAI
errHuang, Lei; Shao, Jialu; Lai, Wenwen; Gu, Hongfeng; Yang, Jieping; Shi, Shi; Wufoyrwoth, Shepherd; Song, Zhe; Zou, Yi; Xu, Yungen; Zhu, Qihua
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Discovery of the novel and potent histamine H1 receptor antagonists for treatment of allergic diseases用于治疗过敏性疾病的新型有效组胺H1受体拮抗剂的发现
err2024-03-01
err1
PREAI
errChu, Zhaoxing; Cen, ab Lifang; Xu, Qinlong; Lin, Gaofeng; Mo, Jiajia; Shao, Li; Zhao, Yan; Li, Jiaming; Ye, Wenfeng; Fang, Tao; Ren, Weijie; Zhu, Qihua; He, Guangwei; Xu, Yungen
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DCLK1 and its oncogenic functions: A promising therapeutic target for cancers
err2024-01-01
err2
PREAI
errYe, Liu; Liu, Beibei; Huang, Jingling; Zhao, Xiaolin; Wang, Yuan; Xu, Yungen; Wang, Shuping
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Discovery of Highly Selective PARP7 Inhibitors with a Novel Scaffold for Cancer Immunotherapy
err2023-12-07
err5
PREAI
errGu, Hongfeng; Yan, Wenxin; Yang, Jieping; Liu, Beibei; Zhao, Xiaolin; Wang, Hongxia; Xu, Wenbo; Wang, Chenghao; Chen, Yang; Dong, Qiuyi; Zhu, Qihua; Xu, Yungen; Zou, Yi
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Discovery of novel dual Bruton's tyrosine kinase (BTK) and Janus kinase 3 (JAK3) inhibitors as a promising strategy for rheumatoid arthritis
err2023-12-01
err4
PREAI
errLiang, Tingting; Cen, Lifang; Wang, Junjie; Cheng, Ming; Guo, Weibo; Wang, Wenjie; Yu, Chunqiu; Zhang, Haifeng; Wang, Yuan; Hao, Zhongyan; Jin, Jiaming; Wu, Yaoyao; Jiang, Teng; Zhu, Qihua; Xu, Yungen
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Design, synthesis and biological evaluation of novel DCLK1 inhibitor containing purine skeleton for the treatment of pancreatic cancer
err2023-12-01
err3
PREAI
errChen, Yuepeng; Meng, Liuqiong; Wang, Wenze; Ye, Liu; Huang, Lei; Wang, Chenghao; Wang, Shuping; Li, Mengyao; Pei, Yingxin; Zhang, Shijie; Zou, Yi; Xu, Yungen
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An overview of limonoid synthetic derivatives as promising bioactive molecules
err2023-11-01
err4
PREAI
errWang, Shaochi; Kuperman, Laura L.; Song, Zhihui; Chen, Yutian; Liu, Kun; Xia, Zongping; Xu, Yungen; Yu, Qiuning
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研究方向

Du, Y.Zou, Y.Niu, J.Cai, Z. Y.Wang, X. N.Qiu, F. H.Yang, G. C.Wu, Y. Z.Xu, Y. G*.靶向蛋白降解肿瘤组织选择性Huang. S. H.Lin. Q. W.Tang. Y. X.Huang. L.Xu. Y. G.*胰腺癌治疗Li, Y.Huang, S. H.Wu, S. Q.Gao, L. L.Sun, Q.Lin, Q. W.Huang, L.Meng, L. Q.Zhu, Q. H*.PARP/BRD4抑制剂He, G. C.Chu, Z. X.Wu, H. H.Wang, J. J.Ge, Y. R.Shen, H.Zhang, S.Shan, J. X.Peng, K. W.Wei, Z. F.IDO1/IDO2双抑制剂癌症免疫治疗Wu. S. Q.Meng. L. Q.Liu. F.Zhu. Q. H.Bai, Y.Jin, J. M.Jiang, T.Ju, Q. R.PARP/PI3K双抑制剂癌症治疗Liu. J. C.Wang. Y.Yang. L.Han. B.Zhang. Y.Bai. Y.Shen. L.Li. M. Y.Jiang. T.Ye. Q. Q.Yu. X. Y.Huang. R. R.Zhang. Z.PARP14通过LPAR5抑制小胶质细胞激活促进卒中后功能恢复Wang. Z. B.Sun. Z. R.Zhang. L.Zhang. W. W.铂基联合疗法Zeng. F. T.Li. X. F.Ran. C. Z.阿尔茨海默病检测Li, H.